Department of Pharmaceutical Chemistry, Manipal College of Pharmaceutical Sciences, Manipal

  • India

Research Output

2020

A Machine Learning Approach for Drug-Target Interaction Prediction using Wrapper Feature Selection and Class Balancing

Redkar, S., Mondal, S., Joseph, A. & Hareesha, K. S., 01-01-2020, (Accepted/In press) In : Molecular Informatics.

Research output: Contribution to journalArticle

2 Citations (Scopus)

Analytical method development using central composite design for estimation of lamotrigine in lipid nanoformulation

Gangurde, P. K., Bhaskaran, N. A., Verma, R., Jose, J. & Kumar, L., 03-2020, In : Materiale Plastice. 57, 1, p. 223-235 13 p.

Research output: Contribution to journalArticle

Open Access
1 Citation (Scopus)

A Review on Anticancer Potentials of Benzothiazole Derivatives

Pathak, N., Rathi, E., Kumar, N., Kini, S. G. & Rao, C. M., 01-01-2020, In : Mini reviews in medicinal chemistry. 20, 1, p. 12-23 12 p.

Research output: Contribution to journalArticle

1 Citation (Scopus)

Asymmetric oxidation of sulfides catalyzed by (R)-6,6'-dibromo-BINOL derived titanium complex

Maddireddy, N. V., Godbole, H. M., Singh, G. P., Kini, S. G. & Shenoy, G. G., 2020, (Accepted/In press) In : Synthetic Communications.

Research output: Contribution to journalArticle

Design, preparation and in vitro characterizations of fluconazole loaded nanostructured lipid carriers

Fernandes, A. V., Pydi, C. R., Verma, R., Jose, J. & Kumar, L., 01-01-2020, In : Brazilian Journal of Pharmaceutical Sciences. 56, e18069.

Research output: Contribution to journalArticle

Open Access
3 Citations (Scopus)

Design, Synthesis, Biological Evaluation and Molecular Dynamic Simulation Studies of Diphenyl Ether Derivatives as Antitubercular and Antibacterial Agents

Khade, A. B., Eshwara, V. K., Boshoff, H. I. M., Arora, K., Tiwari, A., Bhat, P., Tiwari, M. & Shenoy, G. G., 09-01-2020, In : ChemistrySelect. 5, 1, p. 201-210 10 p.

Research output: Contribution to journalArticle

Open Access

Design, synthesis, evaluation, and molecular dynamic simulation of triclosan mimic diphenyl ether derivatives as antitubercular and antibacterial agents

Khade, A. B., Boshoff, H. I. M., Arora, K., Vandana, K. E., Verma, R. & Shenoy, G. G., 01-01-2020, (Accepted/In press) In : Structural Chemistry.

Research output: Contribution to journalArticle

1 Citation (Scopus)

Inhibition performances of spirocyclopropane derivatives for mild steel protection in HCl

Chafiq, M., Chaouiki, A., Lgaz, H., Salghi, R., Bhaskar, K. V., Marzouki, R., Bhat, K. S., Ali, I. H., Khan, M. I. & Chung, I. M., 01-03-2020, In : Materials Chemistry and Physics. 243, 122582.

Research output: Contribution to journalArticle

4 Citations (Scopus)

Is viral E6 oncoprotein a viable target? A critical analysis in the context of cervical cancer

Kumar, A., Rathi, E., Hariharapura, R. C. & Kini, S. G., 01-01-2020, (Accepted/In press) In : Medicinal Research Reviews.

Research output: Contribution to journalReview article

Large-Scale Stereoselective Synthesis of 1,3-Oxathiolane Nucleoside, Lamivudine, via ZrCl4-Mediated N-Glycosylation

Aher, U. P., Srivastava, D., Jadhav, H. S., Singh, G. P., Jayashree, B. S. & Shenoy, G. G., 20-03-2020, In : Organic Process Research and Development. 24, 3, p. 387-397 11 p.

Research output: Contribution to journalArticle

Naringin nano-ethosomal novel sunscreen creams: Development and performance evaluation

Gollavilli, H., Hegde, A. R., Managuli, R. S., Bhaskar, K. V., Dengale, S. J., Reddy, M. S., Kalthur, G. & Mutalik, S., 09-2020, In : Colloids and Surfaces B: Biointerfaces. 193, 111122.

Research output: Contribution to journalArticle

New spirocyclopropane derivatives: synthesis and evaluation of their performances toward corrosion inhibition of mild steel in acidic media

Chafiq, M., Chaouiki, A., Lgaz, H., Salghi, R., Bhaskar, K. V., Thakur, P. S., Bhat, K. S., Ali, I. H., Khan, M. I. & Chung, I. M., 01-01-2020, (Accepted/In press) In : Research on Chemical Intermediates.

Research output: Contribution to journalArticle

1 Citation (Scopus)

Rosuvastatin based novel 3-substituted isocoumarins / 3-alkylidenephthalides: Ultrasound assisted synthesis and identification of new anticancer agents

Kumar, J. S., Thirupataiah, B., Medishetti, R., Ray, A., Bele, S. D., Hossain, K. A., Reddy, G. S., Edwin, R. K., Joseph, A., Kumar, N., Shenoy, G. G., Rao, C. M. & Pal, M., 01-09-2020, In : European Journal of Medicinal Chemistry. 201, 112335.

Research output: Contribution to journalArticle

Structure-based identification of small molecules against influenza A virus endonuclease: an in silico and in vitro approach

K, S. D., Puranik, R., N, S., K, K., Fathima, F., K R, A., Joseph, A., J, A., Arunkumar, G. & Mudgal, P. P., 01-06-2020, In : Pathogens and Disease. 78, 4

Research output: Contribution to journalArticle

Synthesis, biological evaluation and molecular dynamics simulation studies of novel diphenyl ethers

Khade, A. B., Kar, S. S., Cinu Thomas, A., Tiwari, A., Tiwari, M., Vandana, K. E., Bhat, P., Varadaraj Bhat, G. & Shenoy, G. G., 01-01-2020, In : Medicinal Chemistry. 16, 2, p. 256-270 15 p.

Research output: Contribution to journalArticle

Synthesis of 11,12-dihydro benzo[c]phenanthridines via a Pd-catalyzed unusual construction of isocoumarin ring/FeCl3-mediated intramolecular arene-allyl cyclization: First identification of a benzo[c]phenanthridine based PDE4 inhibitor

Thirupataiah, B., Reddy, G. S., Ghule, S. S., Kumar, J. S., Mounika, G., Hossain, K. A., Mudgal, J., Mathew, J. E., Shenoy, G. G., Parsa, K. V. L. & Pal, M., 04-2020, In : Bioorganic Chemistry. 97, 103691.

Research output: Contribution to journalArticle

2019

An improved synthesis of latanoprost involving effective control on 15(S) diastereomer

Sasane, S. A., Bhise, N. B., Singh, G. P., Joseph, A. & Shenoy, G. G., 17-09-2019, In : Synthetic Communications. 49, 18, p. 2350-2356 7 p.

Research output: Contribution to journalArticle

Application of Ugi three component reaction for the synthesis of quinapril hydrochloride

Borase, B. B., Godbole, H. M., Singh, G. P., Upadhyay, P. R., Trivedi, A., Bhat, V. & Shenoy, G. G., 01-01-2019, (Accepted/In press) In : Synthetic Communications.

Research output: Contribution to journalArticle

Open Access

Catalytic asymmetric oxidation of sulfides to sulfoxides using (R)-6,6 -Diphenyl-BINOL as a chiral ligand

Maddireddy, N. V., Godbole, H. M., Singh, G. P., Kini, S. G. & Shenoy, G. G., 01-07-2019, In : Journal of Chemical Sciences. 131, 7, 64.

Research output: Contribution to journalArticle

Cerotato de 1-triacontanol aislado de marsilea quadrifolia linn. Protege las neuronas CA3 del hipocampo y mejora el déficit de memoria especial en ratas epilépticas crónicas

Translated title of the contribution: 1-triacontanol cerotate isolated from marsilea quadrifolia linn. Safeguards hippocampal CA3 neurons and augments special memory deficit in chronic epileptic ratsSnehunsu, A., Nayak, S. B., Kandwal, M., Piyali, A., Adiga, M., Sahoo, P., Medabala, T., Rao, K. R. & Joseph, A., 01-01-2019, In : International Journal of Morphology. 37, 1, p. 265-272 8 p.

Research output: Contribution to journalArticle

Open Access
3 Citations (Scopus)

Design, synthesis, in silico and in vitro evaluation of novel diphenyl ether derivatives as potential antitubercular agents

Tiwari, A. P., Sridhar, B., Boshoff, H. I., Arora, K., Gautham Shenoy, G., Vandana, K. E. & Varadaraj Bhat, G., 01-01-2019, (Accepted/In press) In : Molecular Diversity.

Research output: Contribution to journalArticle

Design, synthesis and evaluation of antitubercular activity of Triclosan analogues

Cinu, T. A., Sidhartha, S. K., Indira, B., Varadaraj, B. G., Vishnu, P. S. & Shenoy, G. G., 01-12-2019, In : Arabian Journal of Chemistry.

Research output: Contribution to journalArticle

Designing of stable co-crystals of zoledronic acid using suitable coformers

Varma, A., Laxmi, P., Pai, A., Pai, G., Vasantharaju, S. G. & Sathyanarayana, M. B., 01-01-2019, In : Chemical and Pharmaceutical Bulletin. 67, 8, p. 816-823 8 p.

Research output: Contribution to journalArticle

Open Access
1 Citation (Scopus)

Enhancement in Dissolution Rate of Atorvastatin Trihydrate Calcium by Formulating Its Porous Tablet Using Sublimation Technique

Singh, S. Y., Salwa, Shirodkar, R. K., Verma, R. & Kumar, L., 01-01-2019, (Accepted/In press) In : Journal of Pharmaceutical Innovation.

Research output: Contribution to journalArticle

4 Citations (Scopus)
6 Citations (Scopus)

Experimental data of fabricated co-crystals of doxorubicin HCl with flavonoids

Laxmi, P., Varma, A., Pai, A. & Sathyanarayana, M. B., 01-07-2019, In : Indian Journal of Pharmaceutical Education and Research. 53, 3, p. S225-S230

Research output: Contribution to journalArticle

Open Access
Open Access

Flavones and their analogues as bioactive compounds – An overview

Jayashree, B. S., Venkatachalam, H. & Mallik, S. B., 01-01-2019, In : Mini-Reviews in Organic Chemistry. 16, 4, p. 377-391 15 p.

Research output: Contribution to journalReview article

1 Citation (Scopus)
3 Citations (Scopus)
6 Citations (Scopus)

InCl 3 mediated heteroarylation of indoles and their derivatization via C[sbnd]H activation strategy: Discovery of 2-(1H-indol-3-yl)-quinoxaline derivatives as a new class of PDE4B selective inhibitors for arthritis and/or multiple sclerosis

Sunke, R., Bankala, R., Thirupataiah, B., Ramarao, E. V. V. S., Kumar, J. S., Doss, H. M., Medishetti, R., Kulkarni, P., Kapavarapu, R. K., Rasool, M., Mudgal, J., Mathew, J. E., Shenoy, G. G., Parsa, K. V. L. & Pal, M., 15-07-2019, In : European Journal of Medicinal Chemistry. 174, p. 198-215 18 p.

Research output: Contribution to journalArticle

4 Citations (Scopus)
1 Citation (Scopus)

In vitro and in vivo anticancer activity of semisynthetic derivatives of betulinic acid

Joseph, A., Srinivasan, K. K., Kutty, N. G., Moorkoth, S., Alex, A. T. & Maliyakkal, N., 01-01-2019, In : Latin American Journal of Pharmacy. 38, 8, p. 1582-1590 9 p.

Research output: Contribution to journalArticle

In vitro antioxidant potential of microbial isolates from diverse habitats

Alex, A. T., Kamath, V., Rao, J. V., Udupa, N. & Joseph, A., 10-2019, In : Research Journal of Pharmacy and Technology. 12, 10, p. 4916-4920 5 p.

Research output: Contribution to journalArticle

L-asparaginase from soil actinomycetes: Optimization of process variables using Plackett Burman method

Kumar, M., Muralidharan, A., Pai, A., Subrahmanyam, V. M. & Kamath, V., 07-2019, In : Research Journal of Pharmacy and Technology. 12, 7, p. 3487-3490 4 p.

Research output: Contribution to journalArticle

Micronutrient and their role in stress related disorders

Samkutty, S., Venkatachalam, H. & Jayashree, B. S., 01-10-2019, In : International Journal of Pharmaceutical Research. 11, 4, p. 902-911 10 p.

Research output: Contribution to journalArticle