Department of Pharmaceutical Chemistry, Manipal College of Pharmaceutical Sciences, Manipal

  • India

Research Output

2012

Effect of ethanol extract of Sphaeranthus indicus on cisplatin-induced nephrotoxicity in rats

Mathew, J. E., Joseph, A., Srinivasan, K., Dinakaran, S. V., Mantri, A. & Movaliya, V., 2012, In : Natural Product Research. 26, 10, p. 933-938 6 p.

Research output: Contribution to journalArticle

5 Citations (Scopus)

Elucidation of Structure-activity Relationship of 2-Quinolone Derivatives and Exploration of Their Antitumor Potential Through Bax-induced Apoptotic Pathway

Kumar, N., Raj, V. P., Jayshree, B. S., Kar, S. S., Anandam, A., Thomas, S., Jain, P., Rai, A. & Rao, C. M., 08-2012, In : Chemical Biology and Drug Design. 80, 2, p. 291-299 9 p.

Research output: Contribution to journalArticle

32 Citations (Scopus)

Superbug NDM-1: A global health problem

Suthar, S. K., Joseph, A., Lohan, S. & Alex, A. T., 2012, In : Der Pharmacia Lettre. 4, 4, p. 1183-1187 5 p.

Research output: Contribution to journalArticle

Synthesis and biological evaluation of novel pyrimidine-2(1H)-ones/thiones as potent anti-inflammatory and anticancer agents

Dinakaran, V. S., Jacob, D. & Mathew, J. E., 2012, In : Medicinal Chemistry Research. 21, 11, p. 3598-3606 9 p.

Research output: Contribution to journalArticle

9 Citations (Scopus)

Synthesis and crystal structure of 4-[2-(Methyl-pyridin2-ylamino)ethoxy]-benzaldoxime

Mahadeva Prasad, T. N., Gaonkar, S. L., Kapoor, K., Gupta, V. K., Shimizu, H., Sridhar, M. A. & Shashidhara Prasad, J., 2012, In : X-ray Structure Analysis Online. 28, 4, p. 25-26 2 p.

Research output: Contribution to journalComment/debate

1 Citation (Scopus)

Synthesis of 3-methylflavones and their antioxidant and antibacterial activities

Jayashree, B. S., Alam, A., Nayak, Y. & Vijay Kumar, D., 08-2012, In : Medicinal Chemistry Research. 21, 8, p. 1991-1996 6 p.

Research output: Contribution to journalArticle

12 Citations (Scopus)
2011

1-(2-Hy-droxy-4-methoxyphenyl)-3-(4-methylphenyl)prop-2-en-1-one

Thippeswamy, G. B., Vijay Kumar, D., Jayashree, B. S., Sridhar, M. A. & Shashidhara Prasad, J., 2011, In : Acta Crystallographica Section E: Structure Reports Online. 67, 4

Research output: Contribution to journalArticle

2 Citations (Scopus)

1-(2-Hy-droxy-5-methyl-phen-yl)-3-(2-methyl-phen-yl)prop-2-en-1-one

Kumar, D. V., Thippeswamy, G. B., Jayashree, B. S. & Sridhar, M. A., 2011, In : Acta Crystallographica Section E: Structure Reports Online. 67, 6

Research output: Contribution to journalArticle

1 Citation (Scopus)

Anti-inflammatory, antipruritic and mast cell stabilizing activity of Aristolochia indica

Mathew, J. E., Kaitheri, S. K., Dinakaranvachala, S. & Jose, M., 01-09-2011, In : Iranian Journal of Basic Medical Sciences. 14, 5, p. 422-427 6 p.

Research output: Contribution to journalArticle

5 Citations (Scopus)

Antimicrobial, antioxidant and in vitro anti-inflammatory activity and phytochemical screening of water extract of wedelia trilobata (L.) hitchc

Govindappa, M., Naga Sravya, S., Poojashri, M. N., Sadananda, T. S., Chandrappa, C. P., Santoyo, G., Sharanappa, P. & Anil Kumar, N. V., 30-10-2011, In : Journal of Medicinal Plant Research. 5, 24, p. 5718-5729 12 p.

Research output: Contribution to journalArticle

16 Citations (Scopus)

Antiulcer activity of leaf extract of lawsonia inermis in albino rats

Goli, V., Macharla, S. P., Vijaya Bhasker, K., Gowrishankar, N. L., Bhaskar, J. & Dhanalakshmi, C., 01-09-2011, In : Research Journal of Pharmacy and Technology. 4, 9, p. 1436-1438 3 p.

Research output: Contribution to journalArticle

4 Citations (Scopus)

Benzothieno[3,2-e][1,2,4]triazolo[4,3-c]pyrimidines: Synthesis, characterization, antimicrobial activity, and incorporation into solid lipid nanoparticles

Panchamukhi, S. I., Mulla, J. A. S., Shetty, N. S., Khazi, M. I. A., Khan, A. Y., Kalashetti, M. B. & Khazi, I. A. M., 06-2011, In : Archiv der Pharmazie. 344, 6, p. 358-365 8 p.

Research output: Contribution to journalArticle

9 Citations (Scopus)

Chemical stability studies of bioadhesive topical gel

Kumar, L. & Verma, R., 01-02-2011, In : International Journal of Pharmacy and Pharmaceutical Sciences. 3, 1, p. 101-104 4 p.

Research output: Contribution to journalArticle

9 Citations (Scopus)
3 Citations (Scopus)

High performance liquid chromatographic determination of carboplatin in injections

Agrawal, G. P., Shenoy, G., Ghosh, A., Bhat, K. & Prabhu, L., 06-10-2011, In : Asian Journal of Chemistry. 23, 11, p. 5095-5098 4 p.

Research output: Contribution to journalArticle

2 Citations (Scopus)

In vitro anticancer activity of microbial isolates from diverse habitats

Treasathomas, A., Venkata Rao, J., Subrahmanyam, V. M., Chandrashekhar, H. R., Maliyakkal, N., Kisan, T. K., Joseph, A. & Udupa, N., 2011, In : Brazilian Journal of Pharmaceutical Sciences. 47, 2, p. 279-287 9 p.

Research output: Contribution to journalArticle

5 Citations (Scopus)

Phytochemical, antioxidant and antimicrobial study of flowers of Nyctanthes arbor-tristis Linn

Srinivasan, K. K., Goomber, A., Kumar, S. S., Thomas, A. T. & Joseph, A., 01-05-2011, In : Pharmacologyonline. 2, p. 16-21 6 p.

Research output: Contribution to journalLetter

2 Citations (Scopus)

Synthesis and crystal structure of 1-(3,5-dichloro-2-hydroxyphenyl)-3-(5- methylfuran-2-yl)prop-2-en-1-one

Thippeswamy, G. B., Vijaykumar, D., Jayashree, B. S., Sridhar, M. A. & Prasad, J. S., 12-09-2011, Solid State Physics - Proceedings of the 55th DAE Solid State Physics Symposium 2010. PART A ed. Vol. 1349. p. 176-177 2 p.

Research output: Chapter in Book/Report/Conference proceedingConference contribution

Synthesis and Crystal Structure of 3-(4-Ethylphenyl)-1-(2-hydroxy-4-methoxyphenyl)prop-2-en-1-one

Thippeswamy, G. B., Vijaykumar, D., Prasad, T. N. M., Jayashree, B. S., Lakshminarayana, B. N., Sridhar, M. A. & Prasad, J. S., 07-11-2011, In : X-ray Structure Analysis Online. 27, 7, p. 39-40 2 p.

Research output: Contribution to journalArticle

1 Citation (Scopus)

Vasorelaxant and antihypertensive effect of Cocos nucifera Linn. endocarp on isolated rat thoracic aorta and DOCA salt-induced hypertensive rats

Bankar, G. R., Nayak, P. G., Bansal, P., Paul, P., Pai, K. S. R., Singla, R. K. & Bhat, V. G., 2011, In : Journal of Ethnopharmacology. 134, 1, p. 50-54 5 p.

Research output: Contribution to journalArticle

33 Citations (Scopus)
2010

1-(2-Hydroxy-5-methylphenyl)-3-(3-methylthiophen-2-yl)prop-2-en-1-one

Thippeswamy, G. B., Vijay Kumar, D., Jayashree, B. S., Sridhar, M. A. & Shashidhara Prasad, J., 2010, In : Acta Crystallographica Section E: Structure Reports Online. 66, 6

Research output: Contribution to journalArticle

3 Citations (Scopus)

2-(2-Chloro-phenoxy)acetohydrazide

Fun, H. K., Quah, C. K., Isloor, A. M., Sunil, D. & Shetty, P., 2010, In : Acta Crystallographica Section E: Structure Reports Online. 66, 1

Research output: Contribution to journalArticle

2 Citations (Scopus)

2-Phenoxy-acetohydrazide

Fun, H. K., Quah, C. K., Isloor, A. M., Sunil, D. & Shetty, P., 2010, In : Acta Crystallographica Section E: Structure Reports Online. 66, 1

Research output: Contribution to journalArticle

6 Citations (Scopus)

Antioxidant and antibacterial activity of new 3-methylflavones

Jayashree, B. S., Alam, A., Kumar, D. V. & Nayak, Y., 01-2010, In : Indian Journal of Heterocyclic Chemistry. 19, 3, p. 237-240 4 p.

Research output: Contribution to journalArticle

4 Citations (Scopus)

Design and synthesis of 2-quinolones as antioxidants and antimicrobials: A rational approach

Jayashree, B. S., Thomas, S. & Nayak, Y., 03-2010, In : Medicinal Chemistry Research. 19, 2, p. 193-209 17 p.

Research output: Contribution to journalArticle

49 Citations (Scopus)

Honey bee sting and venom offering active as well as passive immunization could reduce swine flu pandemic A (H1N1)

Singla, R. K. & Bhat, V. G., 2010, In : Medical Hypotheses. 74, 3, p. 617-618 2 p.

Research output: Contribution to journalArticle

3 Citations (Scopus)
22 Citations (Scopus)

Synthesis, anthelmintic and anti-inflammatory activities of some novel imidazothiazole sulfides and sulfones

Shetty, N. S., Khazi, I. A. M. & Ahn, C., 20-08-2010, In : Bulletin of the Korean Chemical Society. 31, 8, p. 2337-2340 4 p.

Research output: Contribution to journalArticle

13 Citations (Scopus)
67 Citations (Scopus)

Synthesis and antitubercular activity of heterocycle substituted diphenyl ether derivatives

Kini, S. G., Bhat, A., Pan, Z. & Dayan, F. E., 2010, In : Journal of Enzyme Inhibition and Medicinal Chemistry. 25, 5, p. 730-736 7 p.

Research output: Contribution to journalArticle

7 Citations (Scopus)

Synthesis and biological evaluation of 2-phenyl chromen-4-ones for their antioxidant and antimicrobial activity

Srinivasan, K. K., Goomber, A., Kumar, S. S., Thomas, A. T. & Joseph, A., 2010, In : Pharmacologyonline. 3, p. 31-37 7 p.

Research output: Contribution to journalArticle

Synthesis of new PCDA-carbohydrate derivatives

Shetty, N. S., Jeon, J. H. & Ahn, C., 20-10-2010, In : Journal of the Korean Chemical Society. 54, 5, p. 650-652 3 p.

Research output: Contribution to journalArticle

Synthesis of novel flavone acyl esters and correlation of log P value with antioxidant and antimicrobial activity

Jayashree, B. S., Thejaswini, J. C., Nayak, Y. & Kumar, D. V., 2010, In : Asian Journal of Chemistry. 22, 2, p. 1055-1066 12 p.

Research output: Contribution to journalArticle

5 Citations (Scopus)
2009

High-performance thin-layer chromatographic analysis of bicalutamide in bulk drug and liposomes

Subramanian, G. S., Karthik, A., Baliga, A., Musmade, P. & Kini, S., 2009, In : Journal of Planar Chromatography - Modern TLC. 22, 4, p. 273-276 4 p.

Research output: Contribution to journalArticle

6 Citations (Scopus)

High-performance thin-layer chromatographic method for analysis of racecadotril in the bulk drug

Prabu, S. L., Singh, T., Kumar, C. D., Joseph, A. & Srinivasan, K. K., 2009, In : Journal of Planar Chromatography - Modern TLC. 22, 4, p. 277-281 5 p.

Research output: Contribution to journalArticle

In-vitro screening and docking study of fosinopril and its analogs: 2nd International Conference on Biomedical and Pharmaceutical Engineering, ICBPE 2009

Kini, S., Chaudhary, J., Arora, S. & simpleware, B. C. . T. O. A. P., 2009.

Research output: Contribution to conferencePaper

Junjappa-ila annulation: α-oxoketene dithioacetal mediated synthesis of substituted benzotriazoles

Shetty, N. S., Lamani, R. S., Panchamukhi, S. I. & Khazi, I. A. M., 07-2009, In : Journal of Heterocyclic Chemistry. 46, 4, p. 774-777 4 p.

Research output: Contribution to journalArticle

Mast cell stabilizing effects of Sphaeranthus indicus

Mathew, J. E., Srinivasan, K. K., Dinakaran, V. & Joseph, A., 2009, In : Journal of Ethnopharmacology. 122, 2, p. 394-396 3 p.

Research output: Contribution to journalArticle

16 Citations (Scopus)

Synthesis, antiinflammatory and antibacterial activity of novel indolyl-isoxazoles

Panda, S. S., Chowdary, P. V. R. & Jayashree, B. S., 2009, In : Indian Journal of Pharmaceutical Sciences. 71, 6, p. 684-687 4 p.

Research output: Contribution to journalArticle

24 Citations (Scopus)

Synthesis, antitubercular activity and docking study of novel cyclic azole substituted diphenyl ether derivatives

Kini, S. G., Bhat, A. R., Bryant, B., Williamson, J. S. & Dayan, F. E., 2009, In : European Journal of Medicinal Chemistry. 44, 2, p. 492-500 9 p.

Research output: Contribution to journalArticle

71 Citations (Scopus)

Synthesis, invitro and invivo anticancer activity of substituted imidazolones

Pai, A., Singla, R. K., Joseph, A., Kedar, T. & Thomas, A. T., 30-08-2009, In : Pharmacologyonline. 2, p. 933-942 10 p.

Research output: Contribution to journalLetter

Synthesis and antimicrobial activitiy of novel barbituric acid and thiohydantoin derivatives of imidazo [2,1- b][1,3, 4] thiadiazoles

Badiger, N. P., Shetty, N. S., Lamani, R. S. & Khazi, I. A. M., 2009, In : Heterocyclic Communications. 15, 6, p. 433-442 10 p.

Research output: Contribution to journalArticle

5 Citations (Scopus)

Synthesis and antimicrobial activity of some novel thienopyrimidines and triazolothienopyrimidines

Shetty, N. S., Lamani, R. S. & Khazi, I. A. M., 05-2009, In : Journal of Chemical Sciences. 121, 3, p. 301-307 7 p.

Research output: Contribution to journalArticle

50 Citations (Scopus)

Synthesis and antimicrobial studies of novel methylene bridged benzisoxazolyl imidazo[2,1-b][1,3,4]thiadiazole derivatives

Lamani, R. S., Shetty, N. S., Kamble, R. R. & Khazi, I. A. M., 07-2009, In : European Journal of Medicinal Chemistry. 44, 7, p. 2828-2833 6 p.

Research output: Contribution to journalArticle

90 Citations (Scopus)

Synthesis and antitumor activity studies of some new fused 1,2,4-triazole derivatives carrying 2,4-dichloro-5-fluorophenyl moiety

Bhat, K. S., Poojary, B., Prasad, D. J., Naik, P. & Holla, B. S., 12-2009, In : European Journal of Medicinal Chemistry. 44, 12, p. 5066-5070 5 p.

Research output: Contribution to journalArticle

106 Citations (Scopus)

Synthesis of some coumarinyl chalcones of pharmacological interest

Jayashree, B. S., Yusuf, S. & Kumar, D. V., 2009, In : Asian Journal of Chemistry. 21, 8, p. 5918-5922 5 p.

Research output: Contribution to journalArticle

10 Citations (Scopus)
2008

Anti-microbial studies on novel 1,3-oxazolidine analogs

Vachala, D., Mathew, J. E., Panneerselvam, P. & Nagarethinam, S., 2008, In : Pharmacologyonline. 2, p. 192-197 6 p.

Research output: Contribution to journalArticle

1 Citation (Scopus)
3 Citations (Scopus)

Cardioprotective activity of 2-substituted-1,3-oxazolidines on CaCl2-induced arrhythmias in isolated frog heart

Dinakaran, V., Mathew, J. E., Vanathi, M. & Panneerselvam, P., 2008, In : Pharmacologyonline. 2, p. 485-492 8 p.

Research output: Contribution to journalArticle

2 Citations (Scopus)

Imatinib quantification in rat plasma by high performance liquid chromatography with ultra violet detection - An application to preclinical pharmacokinetic study

Shetty, R., Kini, S., Musmade, P., Theerthahalli, A., Mohan, C., Bhat, K. M., Patel, J. & Kumar, V., 2008, In : Pharmacologyonline. 3, p. 752-760 9 p.

Research output: Contribution to journalArticle