Department of Pharmaceutical Chemistry, Manipal College of Pharmaceutical Sciences, Manipal

  • India

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2019
8 Citations (Scopus)

Experimental data of fabricated co-crystals of doxorubicin HCl with flavonoids

Laxmi, P., Varma, A., Pai, A. & Sathyanarayana, M. B., 01-07-2019, In : Indian Journal of Pharmaceutical Education and Research. 53, 3, p. S225-S230

Research output: Contribution to journalArticle

Open Access
Open Access
3 Citations (Scopus)
6 Citations (Scopus)

InCl 3 mediated heteroarylation of indoles and their derivatization via C[sbnd]H activation strategy: Discovery of 2-(1H-indol-3-yl)-quinoxaline derivatives as a new class of PDE4B selective inhibitors for arthritis and/or multiple sclerosis

Sunke, R., Bankala, R., Thirupataiah, B., Ramarao, E. V. V. S., Kumar, J. S., Doss, H. M., Medishetti, R., Kulkarni, P., Kapavarapu, R. K., Rasool, M., Mudgal, J., Mathew, J. E., Shenoy, G. G., Parsa, K. V. L. & Pal, M., 15-07-2019, In : European Journal of Medicinal Chemistry. 174, p. 198-215 18 p.

Research output: Contribution to journalArticle

4 Citations (Scopus)
1 Citation (Scopus)

In vitro and in vivo anticancer activity of semisynthetic derivatives of betulinic acid

Joseph, A., Srinivasan, K. K., Kutty, N. G., Moorkoth, S., Alex, A. T. & Maliyakkal, N., 01-01-2019, In : Latin American Journal of Pharmacy. 38, 8, p. 1582-1590 9 p.

Research output: Contribution to journalArticle

In vitro antioxidant potential of microbial isolates from diverse habitats

Alex, A. T., Kamath, V., Rao, J. V., Udupa, N. & Joseph, A., 10-2019, In : Research Journal of Pharmacy and Technology. 12, 10, p. 4916-4920 5 p.

Research output: Contribution to journalArticle

L-asparaginase from soil actinomycetes: Optimization of process variables using Plackett Burman method

Kumar, M., Muralidharan, A., Pai, A., Subrahmanyam, V. M. & Kamath, V., 07-2019, In : Research Journal of Pharmacy and Technology. 12, 7, p. 3487-3490 4 p.

Research output: Contribution to journalArticle

Micronutrient and their role in stress related disorders

Samkutty, S., Venkatachalam, H. & Jayashree, B. S., 01-10-2019, In : International Journal of Pharmaceutical Research. 11, 4, p. 902-911 10 p.

Research output: Contribution to journalArticle

1 Citation (Scopus)
2 Citations (Scopus)

Novel isatin-indole derivatives as potential inhibitors of chorismate mutase (CM): Their synthesis along with unexpected formation of 2-indolylmethylamino benzoate ester under Pd-Cu catalysis

Reddy, G. S., Hossain, K. A., Kumar, J. S., Thirupataiah, B., Edwin, R. K., Giliyaru, V. B., Chandrashekhar Hariharapura, R., Shenoy, G. G., Misra, P. & Pal, M., 01-01-2019, In : RSC Advances. 10, 1, p. 289-297 9 p.

Research output: Contribution to journalArticle

Open Access

Photodegradation of methylcobalamin and its determination in a commercial formulation

Chamle, A. H., Shane, N. L. J., Pai, A. & Muddukrishna, B. S., 01-01-2019, In : Indian Journal of Pharmaceutical Sciences. 81, 1, p. 57-62 6 p.

Research output: Contribution to journalArticle

Open Access
4 Citations (Scopus)

Solubility enhancement of ticagrelor by co-crystal technology: Preparation, solid state characterization and solubility studies

Shane, N. L. J., Pai, A., Pai, G., Pai, V., Sg, V. & Sathyanarayana, M. B., 01-01-2019, In : Latin American Journal of Pharmacy. 38, 10, p. 2051-2056 6 p.

Research output: Contribution to journalArticle

2 Citations (Scopus)

Synthesis and characterization of novel chiral imidazolium and pyridinium ionic liquids derived from tartaric acid and 2-oxazolidinone

Nehate, S. P., Godbole, H. M., Singh, G. P., Mathew, J. E. & Shenoy, G. G., 03-05-2019, In : Synthetic Communications. 49, 9, p. 1173-1180 8 p.

Research output: Contribution to journalArticle

Synthesis of 3-indolylmethyl substituted (pyrazolo/benzo)triazinone derivatives under Pd/Cu-catalysis: Identification of potent inhibitors of chorismate mutase (CM)

Reddy, G. S., Snehalatha, A. V., Edwin, R. K., Hossain, K. A., Giliyaru, V. B., Hariharapura, R. C., Gautham Shenoy, G., Misra, P. & Pal, M., 01-10-2019, In : Bioorganic Chemistry. 91, 103155.

Research output: Contribution to journalArticle

4 Citations (Scopus)

Targeting HIV-TB coinfection by developing novel piperidin-4-substituted imines: Design, synthesis, in vitro and in silico studies

Kumar, A., Revathi, R., Sriram, D., Curreli, F., Debnath, A. K., Pai, K. S. & Kini, S. G., 01-06-2019, In : Archiv der Pharmazie. 352, 6, 1800358.

Research output: Contribution to journalArticle

2020

A Machine Learning Approach for Drug-Target Interaction Prediction using Wrapper Feature Selection and Class Balancing

Redkar, S., Mondal, S., Joseph, A. & Hareesha, K. S., 01-01-2020, (Accepted/In press) In : Molecular Informatics.

Research output: Contribution to journalArticle

2 Citations (Scopus)

Analytical method development using central composite design for estimation of lamotrigine in lipid nanoformulation

Gangurde, P. K., Bhaskaran, N. A., Verma, R., Jose, J. & Kumar, L., 03-2020, In : Materiale Plastice. 57, 1, p. 223-235 13 p.

Research output: Contribution to journalArticle

Open Access
1 Citation (Scopus)

A Review on Anticancer Potentials of Benzothiazole Derivatives

Pathak, N., Rathi, E., Kumar, N., Kini, S. G. & Rao, C. M., 01-01-2020, In : Mini reviews in medicinal chemistry. 20, 1, p. 12-23 12 p.

Research output: Contribution to journalArticle

1 Citation (Scopus)

Asymmetric oxidation of sulfides catalyzed by (R)-6,6'-dibromo-BINOL derived titanium complex

Maddireddy, N. V., Godbole, H. M., Singh, G. P., Kini, S. G. & Shenoy, G. G., 2020, (Accepted/In press) In : Synthetic Communications.

Research output: Contribution to journalArticle

Design, preparation and in vitro characterizations of fluconazole loaded nanostructured lipid carriers

Fernandes, A. V., Pydi, C. R., Verma, R., Jose, J. & Kumar, L., 01-01-2020, In : Brazilian Journal of Pharmaceutical Sciences. 56, e18069.

Research output: Contribution to journalArticle

Open Access
3 Citations (Scopus)

Design, Synthesis, Biological Evaluation and Molecular Dynamic Simulation Studies of Diphenyl Ether Derivatives as Antitubercular and Antibacterial Agents

Khade, A. B., Eshwara, V. K., Boshoff, H. I. M., Arora, K., Tiwari, A., Bhat, P., Tiwari, M. & Shenoy, G. G., 09-01-2020, In : ChemistrySelect. 5, 1, p. 201-210 10 p.

Research output: Contribution to journalArticle

Open Access

Design, synthesis, evaluation, and molecular dynamic simulation of triclosan mimic diphenyl ether derivatives as antitubercular and antibacterial agents

Khade, A. B., Boshoff, H. I. M., Arora, K., Vandana, K. E., Verma, R. & Shenoy, G. G., 01-01-2020, (Accepted/In press) In : Structural Chemistry.

Research output: Contribution to journalArticle

1 Citation (Scopus)
1 Citation (Scopus)

Inhibition performances of spirocyclopropane derivatives for mild steel protection in HCl

Chafiq, M., Chaouiki, A., Lgaz, H., Salghi, R., Bhaskar, K. V., Marzouki, R., Bhat, K. S., Ali, I. H., Khan, M. I. & Chung, I. M., 01-03-2020, In : Materials Chemistry and Physics. 243, 122582.

Research output: Contribution to journalArticle

6 Citations (Scopus)

Large-Scale Stereoselective Synthesis of 1,3-Oxathiolane Nucleoside, Lamivudine, via ZrCl4-Mediated N-Glycosylation

Aher, U. P., Srivastava, D., Jadhav, H. S., Singh, G. P., Jayashree, B. S. & Shenoy, G. G., 20-03-2020, In : Organic Process Research and Development. 24, 3, p. 387-397 11 p.

Research output: Contribution to journalArticle

Naringin nano-ethosomal novel sunscreen creams: Development and performance evaluation

Gollavilli, H., Hegde, A. R., Managuli, R. S., Bhaskar, K. V., Dengale, S. J., Reddy, M. S., Kalthur, G. & Mutalik, S., 09-2020, In : Colloids and Surfaces B: Biointerfaces. 193, 111122.

Research output: Contribution to journalArticle

1 Citation (Scopus)

New spirocyclopropane derivatives: synthesis and evaluation of their performances toward corrosion inhibition of mild steel in acidic media

Chafiq, M., Chaouiki, A., Lgaz, H., Salghi, R., Bhaskar, K. V., Thakur, P. S., Bhat, K. S., Ali, I. H., Khan, M. I. & Chung, I. M., 01-01-2020, (Accepted/In press) In : Research on Chemical Intermediates.

Research output: Contribution to journalArticle

2 Citations (Scopus)
Open Access

Rosuvastatin based novel 3-substituted isocoumarins / 3-alkylidenephthalides: Ultrasound assisted synthesis and identification of new anticancer agents

Kumar, J. S., Thirupataiah, B., Medishetti, R., Ray, A., Bele, S. D., Hossain, K. A., Reddy, G. S., Edwin, R. K., Joseph, A., Kumar, N., Shenoy, G. G., Rao, C. M. & Pal, M., 01-09-2020, In : European Journal of Medicinal Chemistry. 201, 112335.

Research output: Contribution to journalArticle

Structure-based identification of small molecules against influenza A virus endonuclease: an in silico and in vitro approach

K, S. D., Puranik, R., N, S., K, K., Fathima, F., K R, A., Joseph, A., J, A., Arunkumar, G. & Mudgal, P. P., 01-06-2020, In : Pathogens and Disease. 78, 4

Research output: Contribution to journalArticle

Synthesis, biological evaluation and molecular dynamics simulation studies of novel diphenyl ethers

Khade, A. B., Kar, S. S., Cinu Thomas, A., Tiwari, A., Tiwari, M., Vandana, K. E., Bhat, P., Varadaraj Bhat, G. & Shenoy, G. G., 01-01-2020, In : Medicinal Chemistry. 16, 2, p. 256-270 15 p.

Research output: Contribution to journalArticle

Synthesis of 11,12-dihydro benzo[c]phenanthridines via a Pd-catalyzed unusual construction of isocoumarin ring/FeCl3-mediated intramolecular arene-allyl cyclization: First identification of a benzo[c]phenanthridine based PDE4 inhibitor

Thirupataiah, B., Reddy, G. S., Ghule, S. S., Kumar, J. S., Mounika, G., Hossain, K. A., Mudgal, J., Mathew, J. E., Shenoy, G. G., Parsa, K. V. L. & Pal, M., 04-2020, In : Bioorganic Chemistry. 97, 103691.

Research output: Contribution to journalArticle

2021

Repurposing of existing FDA approved drugs for Neprilysin inhibition: An in-silico study

Sankhe, R., Rathi, E., Manandhar, S., Kumar, A., Pai, S. R. K., Kini, S. G. & Kishore, A., 15-01-2021, In : Journal of Molecular Structure. 1224, 129073.

Research output: Contribution to journalArticle

Open Access