Gautham G Shenoy

An improved synthesis of latanoprost involving effective control on 15(S) diastereomer

Sasane, S. A., Bhise, N. B., Singh, G. P., Joseph, A. & Shenoy, G. G., 17-09-2019, In : Synthetic Communications. 49, 18, p. 2350-2356 7 p.

Research output: Contribution to journal › Article

latanoprost

Hydroxyl Radical

Crystallization

Purification

Application of Ugi three component reaction for the synthesis of quinapril hydrochloride

Borase, B. B., Godbole, H. M., Singh, G. P., Upadhyay, P. R., Trivedi, A., Bhat, V. & Shenoy, G. G., 01-01-2019, (Accepted/In press) In : Synthetic Communications.

Research output: Contribution to journal › Article

Amides

Blood pressure

Pharmaceutical Preparations

quinapril

Catalytic asymmetric oxidation of sulfides to sulfoxides using (R)-6,6 ^′ -Diphenyl-BINOL as a chiral ligand

Maddireddy, N. V., Godbole, H. M., Singh, G. P., Kini, S. G. & Shenoy, G. G., 01-07-2019, In : Journal of Chemical Sciences. 131, 7, 64.

Research output: Contribution to journal › Article

Sulfoxides

Sulfides

Oxidants

Ligands

Oxidation

1 Citation (Scopus)

Design, synthesis, and evaluation of novel diphenyl ether derivatives against drug-susceptible and drug-resistant strains of Mycobacterium tuberculosis

Kar, S. S., Bhat, V. G., Shenoy, V. P., Bairy, I. & Shenoy, G. G., 01-01-2019, In : Chemical Biology and Drug Design. 93, 1, p. 60-66 7 p.

Research output: Contribution to journal › Article

Antitubercular Agents

Phenyl Ethers

Tuberculosis

Derivatives

Vero Cells

3 Citations (Scopus)

Design, Synthesis and Evaluation of Antitubercular Activity of Novel 1,2,4-Triazoles Against MDR Strain of Mycobacterium tuberculosis

Ganesh Kumar, T. N. V., Gautham Shenoy, G., Kar, S. S., Shenoy, V. & Bairy, I., 01-01-2018, In : Pharmaceutical Chemistry Journal. 51, 10, p. 907-917 11 p.

Research output: Contribution to journal › Article

Econazole

Mycobacterium tuberculosis

Antitubercular Agents

Azoles

Mycobacterium

8 Citations (Scopus)

Design, synthesis and evaluation of antitubercular activity of Triclosan analogues

Cinu, T. A., Sidhartha, S. K., Indira, B., Varadaraj, B. G., Vishnu, P. S. & Shenoy, G. G., 2015, In : Arabian Journal of Chemistry.

Research output: Contribution to journal › Article

2 Citations (Scopus)

Development and validation of a new reversed-phase HPLC method for the determination of ezetimibe in pharmaceutical dosage forms

Panjwani, G., Shetty, R., Shenoy, G. & Dhamecha, D., 01-01-2013, In : Indian Journal of Pharmaceutical Education and Research. 47, 1, p. 7-12 6 p.

Research output: Contribution to journal › Article

Dosage Forms

High Pressure Liquid Chromatography

Pharmaceutical Preparations

Anticholesteremic Agents

Enterocytes

Effect of topical recombinant lysostaphin against methicillin resistant staphylococcus aureus infection in a mouse burn wound model

Narasimhaswamy, N., Bairy, I., Musharraf, S., Kumar, S., Nayak, U. Y., Shenoy, G. & Bairy, L. K., 2015, In : International Journal of Pharma and Bio Sciences. 6, 4, p. B1151-B1157

Research output: Contribution to journal › Article

Enantioselective Michael addition of malonic esters to benzalacetophenone by using chiral phase transfer catalysts derived from proline-mandelic acid/tartaric acid

Mahajan, D. P., Godbole, H. M., Singh, G. P. & Shenoy, G. G., 01-07-2019, In : Journal of Chemical Sciences. 131, 7, 67.

Research output: Contribution to journal › Article

Chalcone

Proline

Esters

Catalysts

Malonates

33 Citations (Scopus)

Fabrication, solid state characterization and bioavailability assessment of stable binary amorphous phases of Ritonavir with Quercetin

Dengale, S. J., Hussen, S. S., Krishna, B. S. M., Musmade, P. B., Gautham Shenoy, G. & Bhat, K., 2015, In : European Journal of Pharmaceutics and Biopharmaceutics. 89, p. 329-338 10 p.

Research output: Contribution to journal › Article

Ritonavir

Quercetin

Biological Availability

Solubility

Fourier Transform Infrared Spectroscopy

2 Citations (Scopus)

High performance liquid chromatographic determination of carboplatin in injections

Agrawal, G. P., Shenoy, G., Ghosh, A., Bhat, K. & Prabhu, L., 06-10-2011, In : Asian Journal of Chemistry. 23, 11, p. 5095-5098 4 p.

Research output: Contribution to journal › Article

Carboplatin

Liquids

Dosage Forms

Pharmaceutical Preparations

Quality control

2 Citations (Scopus)

InCl ₃ mediated heteroarylation of indoles and their derivatization via C[sbnd]H activation strategy: Discovery of 2-(1H-indol-3-yl)-quinoxaline derivatives as a new class of PDE4B selective inhibitors for arthritis and/or multiple sclerosis

Sunke, R., Bankala, R., Thirupataiah, B., Ramarao, E. V. V. S., Kumar, J. S., Doss, H. M., Medishetti, R., Kulkarni, P., Kapavarapu, R. K., Rasool, M., Mudgal, J., Mathew, J. E., Shenoy, G. G., Parsa, K. V. L. & Pal, M., 15-07-2019, In : European Journal of Medicinal Chemistry. 174, p. 198-215 18 p.

Research output: Contribution to journal › Article

Indoles

Quinoxalines

Zebrafish

Multiple Sclerosis

Arthritis

9 Citations (Scopus)

Insights on the antioxidant potential of 1, 2, 4-triazoles: Synthesis, screening & QSAR studies

Pokuri, S., Singla, R. K., Bhat, V. G. & Shenoy, G. G., 2014, In : Current Drug Metabolism. 15, 4, p. 389-397 9 p.

Research output: Contribution to journal › Article

In silico studies, synthesis and anticancer activity of novel diphenyl ether-based pyridine derivatives

Verma, R., Bairy, I., Tiwari, M., Bhat, G. V. & Shenoy, G. G., 01-01-2019, In : Molecular Diversity.

Research output: Contribution to journal › Article

Computer Simulation

Pyridine

Ethers

ethers

pyridines

2 Citations (Scopus)

In vitro activity of recombinant lysostaphin in combination with linezolid, vancomycin and oxacillin against methicillin-resistant Staphylococcus aureus

Narasimhaswamy, N., Bairy, I., Shenoy, G. & Bairy, L., 01-08-2017, In : Iranian Journal of Microbiology. 9, 4, p. 208-212 5 p.

Research output: Contribution to journal › Article

Linezolid

Lysostaphin

Oxacillin

Vancomycin

Methicillin-Resistant Staphylococcus aureus

8 Citations (Scopus)

Preparation, solid state characterisation of Paclitaxel and Naringen Cocrystals with improved solubility

Muddukrishna, B. S., Dengale, S. J., Shenoy, G. G. & Bhat, K., 2016, In : International Journal of Applied Pharmaceutics. 8, 4, p. 32-37 6 p.

Research output: Contribution to journal › Article

Paclitaxel

Solubility

Pharmaceutical Preparations

Powder Diffraction

Fourier Transform Infrared Spectroscopy

54 Citations (Scopus)

Preparation and characterization of co-amorphous Ritonavir-Indomethacin systems by solvent evaporation technique: Improved dissolution behavior and physical stability without evidence of intermolecular interactions

Dengale, S. J., Ranjan, O. P., Hussen, S. S., Krishna, B. S. M., Musmade, P. B., Gautham Shenoy, G. & Bhat, K., 01-10-2014, In : European Journal of Pharmaceutical Sciences. 62, p. 57-64 8 p.

Research output: Contribution to journal › Article

Ritonavir

Indomethacin

Solubility

Pharmaceutical Preparations

Technology

1 Citation (Scopus)

Preparation and solid state characterization of paclitaxel cocrystals

Muddukrishna, B. S., Bhat, K. & Shenoy, G. G., 2014, In : Research Journal of Pharmacy and Technology. 7, 1, p. 64-69 6 p.

Research output: Contribution to journal › Article

Paclitaxel

Pharmaceutical Preparations

Solubility

Powder Diffraction

Fourier Transform Infrared Spectroscopy

Production of β -cyclodextrin from pH and thermo stable cyclodextrin glycosyl transferase, obtained from Arthrobacter mysorens and its evaluation as a drug carrier for irbesartan

Rajesh, Y., Narayanan, K., Reddy, M. S., Bhaskar, V. K., Shenoy, G. G., Subrahmanyam, V. M. & Rao, J. V., 2015, In : Current Drug Delivery. 12, 4, p. 444-453 10 p.

Research output: Contribution to journal › Article

2 Citations (Scopus)

Propargylamine (secondary) as a building block in indole synthesis involving ultrasound assisted Pd/Cu-catalyzed coupling-cyclization method: Unexpected formation of (pyrazole)imine derivatives

Sujeevan Reddy, G., Babu Nallapati, S., Sri Saranya, P. S. V. K., Sridhar, B., Bhat Giliyaru, V., Chandrashekhar Hariharapura, R., Gautham Shenoy, G. & Pal, M., 26-12-2018, In : Tetrahedron Letters. 59, 52, p. 4587-4592 6 p.

Research output: Contribution to journal › Article

Indoles

Imines

Cyclization

Ultrasonics

Derivatives

1 Citation (Scopus)

Quantification of sennosides by reverse phase high performance liquid chromatography coupled with electro spray ionization tandem mass spectrometry in Unani formulations

Shreedhara, C. S., Ghosh, A., Shenoy, G., Shetty, R., Kumar, V. S. & Sanghai, D. B., 2013, In : International Journal of Pharmacognosy and Phytochemical Research. 4, 4, p. 124-126 3 p.

Research output: Contribution to journal › Article

Rational design and synthesis of novel diphenyl ether derivatives as antitubercular agents

Kar, S. S., Bhat G, V., Praveen Rao, P. N., vishnu prasad, S., Bairy, I. & Shenoy, G. G., 18-07-2016, In : Drug Design, Development and Therapy. 10, p. 2299-2310

Research output: Contribution to journal › Article

Triclosan

Antitubercular Agents

Mycobacterium tuberculosis

Acyl Carrier Protein

Vero Cells

5 Citations (Scopus)

Rational design and synthesis of novel diphenyl ether derivatives as antitubercular agents

Kar, S. S., Bhat, V. G., Rao, P. P. N., Shenoy, V. P., Bairy, I. & Shenoy, G. G., 18-07-2016, In : Drug Design, Development and Therapy. 10, p. 2299-2310 12 p.

Research output: Contribution to journal › Article

Triclosan

Antitubercular Agents

Mycobacterium tuberculosis

Acyl Carrier Protein

Vero Cells

1 Citation (Scopus)

Response Surface Methodology for Optimization of Ultrasound-Assisted Transdermal Delivery and Skin Retention of Asenapine Maleate

Manikkath, J., Shenoy, G. G., Pandey, S. & Mutalik, S., 01-01-2019, (Accepted/In press) In : Journal of Pharmaceutical Innovation.

Research output: Contribution to journal › Article

Skin

Pharmaceutical Preparations

Bipolar Disorder

Antipsychotic Agents

Biological Availability

Stability indicating HPLC method for venlafaxine hydrochloride capsules

Vijayaraghavan, R., Radha, S., Shenoy Gautham, G., Jain, S., Vaidya, L. & Ahmad, F., 2008, In : Asian Journal of Chemistry. 20, 8, p. 6297-6300 4 p.

Research output: Contribution to journal › Article

Sodium Acetate

Dosage Forms

Capsules

Buffers

Degradation

76 Citations (Scopus)

Structure-activity relationships at the 5-position of thiolactomycin: An intact (5R)-isoprene unit is required for activity against the condensing enzymes from Mycobacterium tuberculosis and Escherichia coli

Kim, P., Zhang, Y. M., Shenoy, G., Nguyen, Q. A., Boshoff, H. I., Manjunatha, U. H., Goodwill, M. B., Lonsdale, J., Price, A. C., Miller, D. J., Duncan, K., White, S. W., Rock, C. O., Barry, C. E. & Dowd, C. S., 12-01-2006, In : Journal of Medicinal Chemistry. 49, 1, p. 159-171 13 p.

Research output: Contribution to journal › Article

Structure-Activity Relationship

Mycobacterium tuberculosis

Catalytic Domain

Escherichia coli

Fatty Acid Synthases

Synthesis, antitubercular evaluation, molecular docking and molecular dynamics studies of 4,6-disubstituted-2-oxo-dihydropyridine-3-carbonitriles

Verma, R., Boshoff, H. I. M., Arora, K., Bairy, I., Tiwari, M., Bhat, V. G. & Shenoy, G. G., 05-12-2019, In : Journal of Molecular Structure. 1197, p. 117-133 17 p.

Research output: Contribution to journal › Article

Triclosan

Molecular dynamics

Docks

Pharmacokinetics

Bacilli

2 Citations (Scopus)

Synthesis, characterization, and preclinical evaluation of new thiazolidin-4-ones substituted with p-chlorophenoxy acetic acid and clofibric acid against insulin resistance and metabolic disorder

Gowdra, V. S., Mudgal, J., Bansal, P., Nayak, P. G., Manohara Reddy, S. A., Shenoy, G. G., Valiathan, M., Chamallamudi, M. R. & Nampurath, G. K., 2014, In : BioMed Research International. 2014, 620434.

Research output: Contribution to journal › Article

Clofibric Acid

Acetic Acid

Insulin Resistance

Insulin

Medical problems

Synthesis, evaluation, molecular docking, and molecular dynamics studies of novel N-(4-[pyridin-2-yloxy]benzyl)arylamine derivatives as potential antitubercular agents

Verma, R., Boshoff, H. I. M., Arora, K., Bairy, I., Tiwari, M., Varadaraj, B. G. & Shenoy, G. G., 01-01-2019, (Accepted/In press) In : Drug Development Research.

Research output: Contribution to journal › Article

Triclosan

Antitubercular Agents

Molecular Dynamics Simulation

Microbial Sensitivity Tests

Bacillus subtilis

15 Citations (Scopus)

Synthesis and antimicrobial activities of 1,3,5 trisubstituted 2-pyrazolines

Gautham Shenoy, G., Bhat, A. R., Varadaraj Bhat, G. & Kotian, M., 2001, In : Indian Journal of Heterocyclic Chemistry. 10, 3, p. 197-200 4 p.

Research output: Contribution to journal › Article

In Vitro Techniques

13 Citations (Scopus)

Synthesis and biological activities of Mannich bases of 7-nitro-2-methyl-4(3H)-quinazolinone

Bhat, A. R., Gautham Shenoy, G. & Kotian, M., 01-04-2000, In : Indian Journal of Heterocyclic Chemistry. 9, 4, p. 319-320 2 p.

Research output: Contribution to journal › Article

Mannich Bases

Bioactivity

2-methyl-4(3H)-quinazolinone

1,3,4-thiadiazole

Synthesis and characterization of novel chiral imidazolium and pyridinium ionic liquids derived from tartaric acid and 2-oxazolidinone

Nehate, S. P., Godbole, H. M., Singh, G. P., Mathew, J. E. & Shenoy, G. G., 03-05-2019, In : Synthetic Communications. 49, 9, p. 1173-1180 8 p.

Research output: Contribution to journal › Article

Oxazolidinones

Ionic Liquids

Sulfides

tartaric acid

Salts

Synthesis and in-vitro antimicrobial activity of 4,6 disubstituted pyrimidines

Bhat, R. & Shenoy, G. G., 2000, In : Pharmacy and Pharmacology Communications. 6, 12, p. 553-557 5 p.

Research output: Contribution to journal › Article

96 Citations (Scopus)

Synthesis and in-vitro antimicrobial activity of new 1,2,4-triazoles

Bhat, A. R., Bhat, G. V. & Shenoy, G. G., 2001, In : Journal of Pharmacy and Pharmacology. 53, 2, p. 267-272 6 p.

Research output: Contribution to journal › Article

Pyrazines

Triazoles

Aspergillus niger

Antitubercular Agents

Antifungal Agents

13 Citations (Scopus)

Synthesis and spectroscopic differentiation of 2- and 4-alkoxythiotetronic acids

Shenoy, G., Kim, P., Goodwin, M., Nguyen, Q. A., Barry, C. E. & Dowd, C. S., 01-03-2004, In : Heterocycles. 63, 3, p. 519-527 9 p.

Research output: Contribution to journal › Article

Ethers

Acids

Alkylation

Ultraviolet spectroscopy

Isomers

Synthesis of 3-indolylmethyl substituted (pyrazolo/benzo)triazinone derivatives under Pd/Cu-catalysis: Identification of potent inhibitors of chorismate mutase (CM)

Reddy, G. S., Snehalatha, A. V., Edwin, R. K., Hossain, K. A., Giliyaru, V. B., Hariharapura, R. C., Gautham Shenoy, G., Misra, P. & Pal, M., 01-10-2019, In : Bioorganic Chemistry. 91, 103155.

Research output: Contribution to journal › Article

Chorismate Mutase

Catalysis

Derivatives

Antitubercular Agents

Cyclization

1 Citation (Scopus)

Synthesis of novel class of 2-oxazolidinone based chiral ionic liquids

Nehate, S. P., Godbole, H. M., Singh, G. P., Mathew, J. E. & Shenoy, G. G., 17-09-2018, In : Synthetic Communications. 48, 18, p. 2435-2440 6 p.

Research output: Contribution to journal › Article

Oxazolidinones

Ionic Liquids

Salts

1 Citation (Scopus)

Synthesis of novel phase transfer catalysts derived from proline-mandelic acid/tartaric acid: their evaluation in enantioselective epoxidation and Darzen condensation

Mahajan, D. P., Godbole, H. M., Singh, G. P. & Shenoy, G. G., 01-03-2019, In : Journal of Chemical Sciences. 131, 3, 22.

Research output: Contribution to journal › Article

Epoxidation

Proline

Condensation

Catalysts

Epoxy Compounds

1 Citation (Scopus)

The: P -toluenesulfonic acid catalyzed single pot synthesis of tetracyclic 1,2-dihydroquinolines: A metal free approach

Hajare, A. K., Jagdale, A. R., Shenoy, G. G. & Sinha, N., 2016, In : New Journal of Chemistry. 40, 6, p. 4888-4890 3 p.

Research output: Contribution to journal › Article

Aniline Compounds

Regioselectivity

Aniline

Cost effectiveness

Ketones

2 Citations (Scopus)

‘One-pot’ organocatalyzed enantioselective synthesis of highly functionalized 3,4,5,6-tetrasubstituted dihydropyrans by sequential Knoevenagel condensation/Michael addition and hemiacetalization

Tilekar, A. R., Jagdale, A. R., Kukreja, G., Shenoy, G. G. & Sinha, N., 2017, In : Tetrahedron Asymmetry. 28, 1, p. 153-161 9 p.

Research output: Contribution to journal › Article

Condensation

condensation

synthesis

Proline

selectivity